Melanotan 1ni peptide ya peptide igereranya yaα-MSH (alpha-melanocyte itera imisemburo). Cyakora nagukora reseptor ya melanocortin-1 (MC1R)kubyutsaumusaruro wa melanin, gutanga bisanzweuruhunagufotora.
Byarabayeyemerewe kuvura erythropoietic protoporphyria (EPP)—Indwara idasanzwe itera kumva cyane izuba. Melanotan 1 ifasha kwiyongerakwihanganira urumuri rwa UV, kugabanyareaction ya Phototoxic, no kuzamurakurinda uruhu kwangirika kwatewe na UV.
GuhitamoMC1R agonist
Yiyongeraumusaruro wa eumelanin
Itangakurinda izuba bisanzwe
GushyigikiraGusana ADN no kurwanya anti-inflammatory
Ibishoboka kurivitiligo, kwirinda kanseri y'uruhu, nakwisiga
Yashakishijwe murikurwanya gusazanaubuvuzi bwa dermatologiya
Isuku ryinshi ≥99%
Synthesis ikomeye ya peptide ikomeye (SPPS)
GMP isa ninganda zikora
Isoko rinini: R&D kurwego rwubucuruzi