komeza kuzamura, kugirango ube igisubizo cyiza ubuziranenge bujyanye nisoko nabaguzi basabwa. Isosiyete yacu ifite gahunda nziza yubwishingizi yashizweho mubyukuri kubiciro byurutonde rwibicuruzwa bitanga ubuziranenge mu BushinwaOrlistatIfu CAS 96829-58-2, “Ubwiza”, “ubunyangamugayo” na “serivisi” nihame ryacu. Ubudahemuka bwacu hamwe nibyo twiyemeje bikomeza kubaha kubitanga. Kora umubonano natwe uyumunsi Kubindi bisobanuro, kora natwe nonaha.
komeza kuzamura, kugirango ube igisubizo cyiza ubuziranenge bujyanye nisoko nabaguzi basabwa. Isosiyete yacu ifite gahunda nziza yubwishingizi yashizweho mubyukuriIfu ya Orlistat, Orlistat, Turizera hamwe na serivisi zacu zihoraho ushobora kubona imikorere myiza kandi igiciro gito muri twe mugihe kirekire. Twiyemeje gutanga serivisi nziza no guha agaciro abakiriya bacu bose. Twizere ko dushobora gushiraho ejo hazaza heza.
| Izina | Leuprorelin |
| Numero ya CAS | 53714-56-0 |
| Inzira ya molekulari | C59H84N16O12 |
| Uburemere bwa molekile | 1209.4 |
| Umubare wa EINECS | 633-395-9 |
| Kuzenguruka byihariye | D25 -31.7 ° (c = 1 muri 1% acide acike) |
| Ubucucike | 1.44 ± 0.1 g / cm3 (Biteganijwe) |
| Imiterere y'ububiko | -15 ° C. |
| Ifishi | Isuku |
| Coefficient ya acide | (pKa) 9.82 ± 0.15 (Biteganijwe) |
| Amazi meza | Gushonga mumazi kuri 1mg / ml |
LH-RHLEUPROLIDE; LEUPROLIDE; LEUPROLIDE (UMUNTU); LEUPRORELIN; [DES-GLY10, D-LEU6, PRO-NHET9] -NHET9) -LUTEINIZINGHORMONE-RELEASINGHORMONE; (DES-GLY10, D-LEU6, PRO-NHET9)
Leuprolide, goserelin, triprelin, na nafarelin ni imiti myinshi ikunze gukoreshwa mu buvuzi kugira ngo ikure intanga ngore zo kuvura kanseri y'ibere mbere yo gucura na kanseri ya prostate. . Ni ukuvuga, gonadotropine isohorwa na pitoito iragabanuka, bigatuma igabanuka rikabije ryimisemburo yimibonano mpuzabitsina isohoka nintanga ngore.
Leuprolide ni imisemburo ya gonadotropine irekura (GnRH), peptide igizwe na acide 9 amine. Iki gicuruzwa kirashobora guhagarika neza imikorere ya sisitemu ya pituito-gonadal, kurwanya imisemburo ya proteolyique no kuba hafi ya reseptor ya GnRH yakira kurusha GnRH, kandi igikorwa cyo guteza imbere irekurwa rya hormone ya luteinizing (LH) nikubye inshuro 20 GnRH. Ifite kandi ingaruka zikomeye zo kubuza imikorere ya pituito-gonad kuruta GnRH. Mu cyiciro cya mbere cyo kuvura, imisemburo itera imisemburo (FSH), LH, estrogene cyangwa androgene irashobora kwiyongera by'agateganyo, hanyuma, kubera kugabanuka kwa glande ya pitoito, gusohora kwa FSH, LH na estrogene cyangwa androgene birabujijwe, bikaviramo gushingira ku misemburo y’imibonano mpuzabitsina. Indwara zishingiye ku gitsina (nka kanseri ya prostate, endometriose, nibindi) zigira ingaruka zo kuvura.
Kugeza ubu, umunyu wa acetate wa leuprolide ukoreshwa cyane cyane mubuvuzi, kubera ko imikorere ya acupate ya leuprolide ihagaze neza mubushyuhe bwicyumba. Amazi agomba gutabwa. Irashobora gukoreshwa mu kuvura imiti ivura endometriose na fibroide yo muri nyababyeyi, ubwangavu bwibanze, kanseri y'ibere mbere yo gucura na kanseri ya prostate, ndetse no kuva amaraso munda ibyara yanduye cyangwa adafite akamaro ko kuvura imisemburo isanzwe. Irashobora kandi gukoreshwa nkuwabanjirije mbere yo kwanga endometrale, ishobora kunaniza endometrium, kugabanya indurwe, no kugabanya ingorane zo kubagwa.komeza gutera imbere, kugirango ube igisubizo cyiza cyo hejuru kijyanye nibisabwa nabaguzi basabwa. Isosiyete yacu ifite gahunda nziza yubwishingizi yashizweho mubyukuri kubiciro byurutonde rwubushinwa Bwiza Bwiza bwo Gutanga Uruganda Urwego rwa Powder CAS 96829-58-2, "Ubwiza", "ubunyangamugayo" na "serivisi" nihame ryacu. Ubudahemuka bwacu hamwe nibyo twiyemeje bikomeza kubaha kubitanga. Kora umubonano natwe uyumunsi Kubindi bisobanuro, kora natwe nonaha.
UrutondeIfu ya Orlistat, Orlistat, Turizera hamwe na serivisi zacu zihoraho ushobora kubona imikorere myiza kandi igura ibicuruzwa bike muri twe mugihe kirekire. Twiyemeje gutanga serivisi nziza no guha agaciro abakiriya bacu bose. Twizere ko dushobora gushiraho ejo hazaza heza.