Ibicuruzwa
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Fmoc-Ile-αMeLeu-Leu-OH
Fmoc-Ile-αMeLeu-Leu-OH ni inyubako ikingira inyubako ya tripeptide ikingira igizwe na α-methylated leucine, ikoreshwa cyane mugushushanya imiti ya peptide kugirango iteze imbere metabolike no guhitamo reseptor.
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Dodecyl Phosphocholine (DPC)
Dodecyl Phosphocholine (DPC) ni intungamubiri ya zwitterionic ikoreshwa cyane mubushakashatsi bwa poroteyine ya membrane na biologiya yubatswe, cyane cyane muri NMR spectroscopy na kristu.
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N-Acetylneuraminic Acide (Neu5Ac Acide Sialic)
Acide N-Acetylneuraminic (Neu5Ac), izwi cyane nka acide sialic, ni monosaccharide isanzwe ibaho igira uruhare mubikorwa bikomeye bya selile na immunite. Ifite uruhare runini mukumenyekanisha ingirabuzimafatizo, kurinda indwara ya patogene, no gukura mu bwonko.
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Ergothioneine
Ergothioneine ni ibintu bisanzwe biboneka muri aside irike ikomoka kuri antioxydants, yizwe kubera imbaraga za cytoprotective na anti-gusaza. Ihindurwamo ibihumyo na bagiteri kandi ikusanyiriza mu ngingo zihura na stress ya okiside.
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NMN
Ubushakashatsi bwibanze kandi bwambere bwabantu bwerekana ko NMN ishobora guteza imbere kuramba, kwihangana kumubiri, no kumenya ubwenge.
Ibiranga API:
Isuku ryinshi ≥99%
Urwego rwa farumasi, rukwiranye numunwa cyangwa inshinge
Yakozwe munsi yuburinganire bwa GMP
NMN API nibyiza gukoreshwa muburyo bwo kurwanya gusaza, kuvura metabolike, nubushakashatsi burambye.
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Glucagon
Glucagon ni imisemburo ya peptide isanzwe ikoreshwa nk'ubuvuzi bwihutirwa bwo kuvura hypoglycemia ikabije kandi yize ku ruhare rwayo mu kugenzura metabolike, kugabanya ibiro, no gusuzuma igifu.
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Motixafortide
Motixafortide ni peptide ya CXCR4 ya antagonist peptide yakozwe kugirango ikangurire ingirabuzimafatizo ya hematopoietic stem selile (HSCs) kugirango ihindurwe autologique kandi iri no kwigwa muri oncology na immunotherapy.
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Glepaglutide
Glepaglutide nikigereranyo kirekire GLP-2 ikora kugirango ivurwe syndrome ngororamubiri ngufi (SBS). Itezimbere amara no gukura, ifasha abarwayi kugabanya gutungwa nimirire yababyeyi.
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Elamipretide
Elamipretide ni tetrapeptide yibasiwe na mitochondria yakozwe mu kuvura indwara ziterwa n'imikorere mibi ya mitochondrial, harimo na myopathie primaire mitochondial, syndrome ya Barth, no kunanirwa k'umutima.
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Donidalorsen
Donidalorsen API ni antisense oligonucleotide (ASO) iri gukorwaho iperereza kugirango ivure umurage wa angioedema (HAE) hamwe nindwara ziterwa na inflammatory. Yizwe murwego rwa RNA igamije kuvura, igamije kugabanya imvugo yaplasma prekallikrein(KLKB1 mRNA). Abashakashatsi bifashisha Donidalorsen kugira ngo basuzume uburyo bwo gucecekesha gene, imiti iterwa na farumasi, no kugenzura igihe kirekire kurwanya indwara ya bradykinin.
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Fitusiran
Fitusiran API ni sintetike ntoya yivanga RNA (siRNA) yakozweho iperereza cyane cyane mubijyanye na hemofilia n'indwara ya coagulation. Ireba iantithrombine (AT cyangwa SERPINC1)gene mu mwijima kugirango igabanye umusaruro wa antithrombine. Abashakashatsi bifashisha Fitusiran kugira ngo basuzume uburyo RNA yivanga (RNAi), gucecekesha gene yihariye y’umwijima, hamwe n’ingamba zo kuvura udushya zo kongera guhuza imitsi mu barwayi ba hémofilia A na B, hamwe na inhibitor.
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Givosiran
Givosiran API ni sintetike ntoya yivanga RNA (siRNA) yize kugirango ivure poropiya ikaze ya hepatike (AHP). Ireba cyane cyaneALAS1gene (aminolevulinic aside synthase 1), igira uruhare munzira ya heme biosynthesis. Abashakashatsi bifashisha Givosiran kugira ngo bakore iperereza ku buvuzi bwa RNA (RNAi) bushingiye ku buvuzi, gucecekesha gene igamije umwijima, no guhindura inzira za metabolike zigira uruhare muri porphiriya n'indwara zishingiye ku ngirabuzima fatizo.