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Igiciro cyasubiwemo Ubushinwa Byuzuye Ubushinwa Kubura Kasi 96829-58-298-2Lk

Ibisobanuro bigufi:

Umubare wa CAB: 96829-58-28-25-28-2

Formulaire ya moleCure: c29h53no5

Uburemere bwa molekile: 495.73

EINIONCs Umubare: 639-755-1

Guhinduranya umwihariko: D20-32.0 ° (C = 1Inchloroform)

Ingingo itetse: 615.9 ± 30.0 ° C (byahanuwe)

Ubucucike: 0.976 ± 0.06G / CM3 (byahanuwe)

Imiterere yo kubika: 2-8 ° C.

 


Ibisobanuro birambuye

Ibicuruzwa

Gutsimbarara ku myizerere ya "Gukora ibintu byo hejuru no guteza inshuti hamwe nabantu muri iki gihe kwisi", mubisanzwe dushyira inyungu zabaguzi mu kigo cyambere cyo gutakaza ubushinwaOrlistat, Kubera ko hashyirwaho imbere mu ntangiriro ya za 90, ubu twubaka umuyoboro wo kugurisha muri Amerika, Ubudage, Aziya, n'ibihugu byinshi byo mu gihugu. Dufite intego yo kubona amasomo yo hejuru yo kuzenguruka isi kandi nyuma yaho!
Kwizirika ku myizerere ya "Gukora ibintu byo hejuru no guteza inshuti hamwe nabantu muri iki gihe baturutse kwisi", mubisanzwe dushyira inyungu z'abaguzi mu mwanya wa mbere kuriUbushinwa 96829-58-28-28-2, Orlistat, Hamwe na leta-yubuhanzi bworoshye bwo gutanga ibitekerezo hamwe nabakozi 300 b'abahanga mu by'ubuhanga, Isosiyete yacu ifite ibisubizo by'ubwoko bwose kuva mu masomo yo hejuru, icyiciro giciriritse kugeza mu cyiciro gito. Ibi byose guhitamo ibintu byiza bitanga abakiriya bacu guhitamo bitandukanye. Byongeye kandi, sosiyete yacu ifata igiciro cyiza kandi cyumvikana, kandi natwe turaguha serivisi nziza oem kubirango byinshi bizwi.

Ibisobanuro birambuye

Izina Leprorelin
Umubare wa Cas 53714-56-0
Formulala C59H84N16O12
Uburemere bwa molekile 1209.4
Umubare wa EINECS 633-395-9
Kuzunguruka D25 -31.7 ° (C = 1 muri 1% acide acide)
Ubucucike 1.44 ± 0.1 g / cm3 (byahanuwe)
Imiterere -15 ° C.
Ifishi Neat
Coeffity (PKA) 9.82 ± 0.15 (byahanuwe)
Amazi Gushonga mumazi kuri 1mg / ml

Synonyme

LH-RHLLEUPLANDE; Leuplide; Leuprol (Umuntu); Leuprorelin; -Nhet9) -Luriinisehormone-Kurekura; (des-gly10, D-leu6, Pros-Gly

Ingaruka ya farumasi

Leuprolide, Goserelin, na Nafarelin, ni ibiyobyabwenge byinshi bikunze gukoreshwa mumyitozo ngororamubiri kugira ngo ukureho intanga ngorerere intanga ngorerere premenopausa na kanseri ya prostate. . Ni ukuvuga, Gonadopropin isohoka na mitoire igabanuka, biganisha ku kugabanuka kwinshi mu misemburo yimibonano mpuzabitsina ihinduka na ovary.

Leuprolide ni Gonmone ya Gonadopropin-kurekura (GNRH) Analog, Peptade igizwe na 9 amino. Iki gicuruzwa kirashobora kubuza neza imikorere ya sisitemu ya Pitoitary-Gonaday, irwanya imisatsi ya Protomeriya hamwe na GNRH Reseptor irusha GNRH, nigikorwa cyo guteza imbere irekurwa rya luteine ​​(lh) rifite inshuro 20 za GNR. Ifite kandi ingaruka zikomeye zibangamira imikorere ya pituitary-gonad kuruta gnrh. Mu cyiciro cyambere cyo kuvura, Folticle gitera imisemburo (Fsh), LH, Estrogene cyangwa na Anderogen irashobora kwiyongera kw'igihe gito, kandi, kubera ko yagabanijwe by'agateganyo, hanyuma, kandi estrogene cyangwa na estrogen cyangwa na Estrogen cyangwa na Estrogen cyangwa bo muri Estrogen cyangwa bongere babuza kwishingikiriza kuri hormone igitsina. Indwara zimibonano mpuzabitsina (nka kanseri ya prostate, endometriose, nibindi) zifite ingaruka zumuco.

Kugeza ubu, umunyu wa acetate wo kwibeshye ukoreshwa cyane cyane ubuvuzi, kuko imikorere ya acetate ihamye ikaze ku bushyuhe bwicyumba. Amazi agomba gutabwa. Irashobora gukoreshwa mugutunganya ibiyobyabwenge bya endometriose na febroide ya nyababyeyi, kanseri yibanze yibanze, kanseri ya premonausal na kanseri ya prostate, ndetse no kuvanga inganda zikora neza cyangwa bidahwitse kumivugo isanzwe. Irashobora kandi gukoreshwa nkiyicye mbere yo gutabwa endometrial, bishobora kuba byoroheje, tugagabanya ingorane zabaguzi mu kigo cyanditseho ubushinwa. Ctilistat orlistat, kuva hashyirwe imbere mu ntangiriro ya za 90, ubu turimo twubaka umuyoboro wo kugurisha muri Amerika, Ubudage, Aziya, n'ibihugu byinshi byo hagati. Dufite intego yo kubona amasomo yo hejuru yo kuzenguruka isi kandi nyuma yaho!
Igiciro cyavuzwe kuriUbushinwa 96829-58-28-28-2. Ibi byose guhitamo ibintu byiza bitanga abakiriya bacu guhitamo bitandukanye. Byongeye kandi, sosiyete yacu ifata igiciro cyiza kandi cyumvikana, kandi natwe turaguha serivisi nziza oem kubirango byinshi bizwi.


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