| Izina | Ifu ya Tirzepatide |
| Isuku | 99% |
| Kugaragara | Ifu yera ya Lyofilize |
| Ubuyobozi | Gutera inshinge |
| Ingano | 10mg, 15mg, 20mg, 30mg |
| Amazi | 3.0% |
| Inyungu | Kuvura diyabete, kunoza igenzura ry'isukari mu maraso |
Tirzepatide ni igitabo gishya cya glucose iterwa na insulineotropique polypeptide / glucagon imeze nka peptide 1 (GLP-1) reseptor agonist yemewe muri Amerika nk'umugereka w'imirire n'imyitozo ngororamubiri kugira ngo igabanye indwara ya glycemic ku bantu bakuze barwaye diyabete yo mu bwoko bwa 2 kandi irimo gukorwaho iperereza kugira ngo ikoreshwe mu gucunga ibiro bidakira, ibintu bikomeye biterwa n'indwara z'umutima ndetse no gucunga indwara ziterwa na virusi. Icyiciro cya 3 SURPASS 1-5 gahunda yo kugerageza ivuriro yateguwe hagamijwe gusuzuma imikorere n’umutekano bya tirzepatide yatewe inshuro imwe mu cyumweru (5, 10 na 15 mg), nka mitiweli cyangwa ivura imiti, mu bantu benshi barwaye diyabete yo mu bwoko bwa 2. Gukoresha tirzepatide mu bushakashatsi bw’ubuvuzi byajyanye no kugabanuka kugaragara kwa gemoglobine glycated (-1.87 kugeza -2.59%, -20 kugeza kuri 28 mmol / mol) hamwe nuburemere bwumubiri (-6.2 kugeza -12.9 kg), ndetse no kugabanya ibipimo bikunze kuba bifitanye isano n’impanuka ziterwa n’umutima nk’umuvuduko wamaraso, umuvuduko ukabije w’amaraso. Tirzepatide yarihanganiye neza, ifite ibyago bike byo kurwara hypoglycaemia mugihe ikoreshejwe idafite insuline cyangwa insuline ya insuline kandi ikerekana umwirondoro wumutekano usa nicyiciro cya GLP-1 reseptor agonist. Kubera iyo mpamvu, ibimenyetso bivuye muri ibyo bigeragezo bivura byerekana ko tirzepatide itanga amahirwe mashya yo kugabanya neza gemoglobine glycated hamwe nuburemere bwumubiri kubantu bakuze barwaye diyabete yo mu bwoko bwa 2.