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Glucagon

Ibisobanuro bigufi:

Glucagon ni imisemburo ya peptide isanzwe ikoreshwa nk'ubuvuzi bwihutirwa bwo kuvura hypoglycemia ikabije kandi yize ku ruhare rwayo mu kugenzura metabolike, kugabanya ibiro, no gusuzuma igifu.


Ibicuruzwa birambuye

Ibicuruzwa

Glucagon API

Glucagon ni imisemburo ya peptide isanzwe ikoreshwa nk'ubuvuzi bwihutirwa bwo kuvura hypoglycemia ikabije kandi yize ku ruhare rwayo mu kugenzura metabolike, kugabanya ibiro, no gusuzuma igifu.

 

Urwego & Ubushakashatsi:

Glucagon ihuza reseptor ya glucagon (GCGR) mu mwijima, itera:

Glycogene isenyuka kugirango glucose yongere amaraso

Lipolysis no gukangurira ingufu

Gastrointestinal motulation modulation (ikoreshwa muri radiologiya)

Irimo gushakishwa kandi mubyibushye, diyabete yo mu bwoko bwa 2, hamwe nubuvuzi bubiri / butatu bwa agonist hamwe na GLP-1 na GIP.

 

Ibiranga API (Itsinda rya Gentolex):

Peptide-yera cyane (≥99%)

Yakozwe hifashishijwe synthesis ya peptide ikomeye (SPPS)

Ubwiza busa na GMP

Bikwiranye ninshinge nibikoresho byihutirwa

Glucagon API ningirakamaro mugutabara hypoglycemia, kwerekana amashusho, hamwe nubushakashatsi bwindwara ya metabolike.


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