Hexarelinni ihurirogukura imisemburo secretagogue peptide (GHS)kandi ikomeyeGHSR-1a agonist, byakozwe kugirango bikangureimisemburo ikura ya endogenous (GH) irekura. Ni iumuryango wa ghrelinkandi igizwe na aside amine esheshatu (hexapeptide), itanga imbaraga zo guhindagurika kwa metabolike hamwe ningaruka zikomeye zo kurekura GH ugereranije nibigereranyo nka GHRP-6.
Hexarelin yizwe cyane kubikorwa byayo muriendocrinology, guta imitsi, gusana umutima, hamwe no kurwanya gusaza, bitewe nubushobozi bwayo busanzwe bwo kuzamura GH nainsuline imeze nkikura 1 (IGF-1)urwego utabanje kwinjiza imisemburo yo hanze.
Hexarelin ihuza naimikurire ya hormone secretagogue reseptor (GHSR-1a)kuri pituito na hypothalamus, bigana ibikorwa byaghrelin- inzara isanzwe yumubiri hamwe na hormone irekura GH.
Ibikorwa by'ingenzi bifatika:
Ikangura pulsatile GH irekura
Yongera kuzengurukaIGF-1urwego
Guteza imbereingaruka za anabolike(gukura kw'imitsi, gukira)
Gushyigikiraibinurenakuvugurura ingirabuzimafatizo
Gicurasi irashobora kwerekanaumutimanaanti-apoptoticIngaruka
Bitandukanye nizindi peptide ya GHS, Hexarelin arabikorantabwo byongera cyane cortisol cyangwa prolactine, gutanga umwirondoro wa endocrine isukuye.
Guteza imbereumubiri unanutseiterambere
Gutezimberegusana imitsi no kuvugurura
Yizesarcopenia, cachexia, hamwe no gukira nyuma yo kubagwa
Ubushakashatsi bwibanze bwerekanakunoza imikorere yumutimanyuma yo gukomeretsa myocardial
Kugabanyafibrosis yumutimakandi ikazamuraibumoso bwo gusohora igice
Ibishobora gukoreshwa murikunanirwa k'umutimanagusaza k'umutimaicyitegererezo
Yiyongeralipolysiskandi aratera imbereinsuline
Gushyigikiraimiti yo kurwanya gusazabinyuze muri GH / IGF-1 gutera imbaraga
Turashobora gufasha kubungabungaubwinshi bwamagufwa nubuzima bufatanije
Isuku ≥ 99%
Byakozwe binyuzesynthesis ikomeye ya peptide (SPPS)
Ibipimo bisa na GMP, endotoxine nkeya hamwe nibisigara bya solvent
Isoko ryoroshye:R&D kurwego rwubucuruzi