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Hexarelin

Ibisobanuro bigufi:

Hexarelin ni imisemburo ikura ya hormone secretagogue peptide (GHS) hamwe na GHSR-1a agonist ikomeye, yakozwe kugirango itume imisemburo ikura ya endogenous ikura (GH). Ni iy'umuryango wigana ghrelin kandi igizwe na acide esheshatu za amine (hexapeptide), itanga imbaraga zo guhinduranya metabolike hamwe ningaruka zikomeye zo kurekura GH ugereranije n’ibigereranyo byabanje nka GHRP-6.

Ibiranga API:

Isuku ≥ 99%

Yakozwe hifashishijwe synthesis ya peptide ikomeye (SPPS)

Ibipimo bisa na GMP, endotoxine nkeya nibisigara bya solvent

Isoko ryoroshye: R&D kurwego rwubucuruzi


Ibicuruzwa birambuye

Ibicuruzwa

Hexarelin API - Incamake y'ibicuruzwa

Hexarelinni ihurirogukura imisemburo secretagogue peptide (GHS)kandi ikomeyeGHSR-1a agonist, byakozwe kugirango bikangureimisemburo ikura ya endogenous (GH) irekura. Ni iumuryango wa ghrelinkandi igizwe na aside amine esheshatu (hexapeptide), itanga imbaraga zo guhindagurika kwa metabolike hamwe ningaruka zikomeye zo kurekura GH ugereranije nibigereranyo nka GHRP-6.

Hexarelin yizwe cyane kubikorwa byayo muriendocrinology, guta imitsi, gusana umutima, hamwe no kurwanya gusaza, bitewe nubushobozi bwayo busanzwe bwo kuzamura GH nainsuline imeze nkikura 1 (IGF-1)urwego utabanje kwinjiza imisemburo yo hanze.


Uburyo bwibikorwa

Hexarelin ihuza naimikurire ya hormone secretagogue reseptor (GHSR-1a)kuri pituito na hypothalamus, bigana ibikorwa byaghrelin- inzara isanzwe yumubiri hamwe na hormone irekura GH.

Ibikorwa by'ingenzi bifatika:

  • Ikangura pulsatile GH irekura

  • Yongera kuzengurukaIGF-1urwego

  • Guteza imbereingaruka za anabolike(gukura kw'imitsi, gukira)

  • Gushyigikiraibinurenakuvugurura ingirabuzimafatizo

  • Gicurasi irashobora kwerekanaumutimanaanti-apoptoticIngaruka

Bitandukanye nizindi peptide ya GHS, Hexarelin arabikorantabwo byongera cyane cortisol cyangwa prolactine, gutanga umwirondoro wa endocrine isukuye.


Ubushakashatsi hamwe nubuvuzi bushoboka

1. Gukura kw'imitsi & Kugarura

  • Guteza imbereumubiri unanutseiterambere

  • Gutezimberegusana imitsi no kuvugurura

  • Yizesarcopenia, cachexia, hamwe no gukira nyuma yo kubagwa

2. Kurinda umutima

  • Ubushakashatsi bwibanze bwerekanakunoza imikorere yumutimanyuma yo gukomeretsa myocardial

  • Kugabanyafibrosis yumutimakandi ikazamuraibumoso bwo gusohora igice

  • Ibishobora gukoreshwa murikunanirwa k'umutimanagusaza k'umutimaicyitegererezo

3. Ibinure binini & Kurwanya gusaza

  • Yiyongeralipolysiskandi aratera imbereinsuline

  • Gushyigikiraimiti yo kurwanya gusazabinyuze muri GH / IGF-1 gutera imbaraga

  • Turashobora gufasha kubungabungaubwinshi bwamagufwa nubuzima bufatanije


Ibiranga API (Itsinda rya Gentolex)

  • Isuku ≥ 99%

  • Byakozwe binyuzesynthesis ikomeye ya peptide (SPPS)

  • Ibipimo bisa na GMP, endotoxine nkeya hamwe nibisigara bya solvent

  • Isoko ryoroshye:R&D kurwego rwubucuruzi


  • Mbere:
  • Ibikurikira:

  • Andika ubutumwa bwawe hano hanyuma utwohereze