Ipamorelin

Ipamorelin API

Ipamorelin ni imisemburo ikura ya pentapeptide ikura ya peptide (GHRP) igizwe na aside amine atanu (Aib-His-D-2-Nal-D-Phe-Lys-NH₂). Nibintu byatoranijwe GHSR-1a agonist ifite ubushobozi bwo gukangura imisemburo ikura (GH) ifite umwihariko. Ugereranije na GHRP zabanje (nka GHRP-2 na GHRP-6), Ipamorelin yerekana guhitamo neza, umutekano ndetse no guhagarara kwa farumasi bitagize ingaruka zikomeye kurwego rwizindi misemburo nka cortisol, prolactine cyangwa ACTH.

Nka peptide yubahwa cyane, Ipamorelin kuri ubu ikoreshwa cyane mubushakashatsi bwo kurwanya gusaza, gusubiza mu buzima busanzwe siporo, gutabara osteoporose, gukira nyuma yo kubagwa no kugenzura imikorere ya metabolike.

Ubushakashatsi hamwe nuburyo bukoreshwa

Ipamorelin iteza imbere kurekura imisemburo ikura ya endogenous (GH) muri pitoito yimbere muguhitamo gukora imisemburo ikura ya hormone ikura (GHSR-1a) no kwigana ibikorwa bya ghrelin. Uburyo bukuru bwa farumasi burimo:
1. Kangura ururenda rwa GH
Ipamorelin ihitamo cyane GHSR-1a, bigatuma glande ya pitoito irekura GH itagize ingaruka zikomeye kurwego rwa ACTH cyangwa cortisol, kandi ifite umutekano mwiza wa endocrine.
2. Kongera intungamubiri za poroteyine no gusana selile
Mu kongera urwego rwa IGF-1, ruteza imbere imitsi ya anabolisme yimitsi, ikongera gusana ingirabuzimafatizo no kuvugurura, kandi ikwiriye gusana ihahamuka, kubagwa no kubaga no kuvura imitsi.
3. Kunoza metabolisme no gukwirakwiza ibinure
GH ifite ingaruka zo gukangurira ibinure no kunoza insuline. Ipamorelin irashobora gufasha mukugenzura imiterere ya metabolike kandi ikoreshwa mubushakashatsi kuri syndrome de metabolike no kuvura umubyibuho ukabije.
4. Kunoza ubwinshi bwamagufwa no kurwanya gusaza
GH / IGF-1 axis irashobora guteza imbere amagufwa no kugabanuka. Ipamorelin yerekana amasezerano muri anti-osteoporose, kuvugurura imvune no kurwanya gusaza.
5. Kunoza injyana ya circadian no gusinzira neza
Kurekura GH mubisanzwe biherekejwe no gusinzira cyane. Ubushakashatsi bwerekanye ko Ipamorelin ishobora kuzamura mu buryo butaziguye imiterere y'ibitotsi no kongera ubushobozi bwo gukira umubiri.
Ubushakashatsi bwibanze no kugenzura neza

Nubwo bikiri mubyiciro byubuvuzi / kare, Ipamorelin yerekanye umutekano mwiza ningirakamaro mubikoko hamwe nubushakashatsi bwabantu:

Urwego rwa GH rwiyongereye cyane (impinga muminota 30, rumara amasaha menshi)

Nta ngaruka igaragara ya cortisol cyangwa pro-ACTH, ingaruka za endocrine zirashobora kugenzurwa

Kunoza imitsi n'imbaraga (cyane cyane mubyitegererezo by'inyamaswa zishaje)

Kunoza nyuma yo gukira no kwihuta gusana

Kwiyongera kurwego rwa IGF-1 bifasha gusana selile no gusubiza antioxydeant

Byongeye kandi, Ipamorelin ifatanije nandi mimetike ya GHRH (nka CJC-1295) mubushakashatsi bumwe bwerekanye ingaruka zoguhuza, bikarushaho kongera imbaraga zo gusohora kwa GH.
Umusaruro wa API nubwishingizi bufite ireme

Ipamorelin API itangwa na Groupe yacu ya Gentolex yateguwe hifashishijwe uburyo bwo hejuru bwa ** bukomeye bwa peptide ya peptide synthesis (SPPS) **, kandi isukuwe neza kandi yipimishije ubuziranenge, ikwiranye nubushakashatsi bwa siyansi niterambere ndetse no gukoresha imiyoboro hakiri kare yimiti yimiti.

Ibicuruzwa birimo:

Isuku ≥99% (ikizamini cya HPLC)
Nta endotoxine, ibisigara bike bisigaye, ibyuma bike ion yanduye
Tanga urutonde rwuzuye rwinyandiko zujuje ubuziranenge: COA, raporo yo kwiga ituze, isesengura ryanduye, nibindi.
Guhindura gram-urwego ~ kilo-urwego rwo gutanga