Izina | Ru-58841 |
Umubare wa Cas | 154992-24-2 |
Formulala | C17H18F3N3NO3 |
Uburemere bwa molekile | 369.34 |
Umubare wa EINECS | 1592732-453-0 |
Ingingo itetse | 493.6 ± 55.0 ° C (byahanuwe) |
Ubucucike | 1.39 |
Imiterere | Yashyizweho ikimenyetso cyumye, ububiko muri firigo, munsi ya -20 ° C. |
Ifishi | Ifu |
Ibara | Cyera |
Gupakira | Pe Umufuka + Umufuka wa Aluminium |
Ru58841; 4- (4,4-Dimeithyl-2,5-Dioxyo-3- nitrile; Onitrile; 4- (3- hydroxybutyl) -4,4-Dimethyl-2,5-Dioxooimidazolididin-1-YL] -2- (Trifluoromethyyl) Ben Zonitrile; ru-58841E: Candyli (kuri) kwihuta (akadomo) com; cs-638; ru58841; ru-58841
Ibisobanuro
Ru 58841 (PSK-3841) ni bondeddor ba Anagoni ba Anagononite iteza imbere imisatsi.Ru58841 ni ibiyobyabwenge by'iperereza byashyizweho kugira ngo bivure Androgenic Alopecia, bizwi kandi ku izina ry'umugabo (MPD).
Nkibintu byingenzi birwanya nandero, ihame ryibikorwa ntabwo rimeze nkibyinshi. Gusaba inyungu zikorwa muburyo butaziguye 5α kugabanuka, kubuza ihinduka rya testosterone muri DHT, kandi rigabanya ibikubiye muri Dht mumubiri. Ru58841 ihagarika umubano hagati yinkuro hamwe numusatsi wa resile, ntabwo bigabanya ibintu bya dht, ariko bigabanya agaciro ka dht hamwe nintego yo kuvura androGanetic alopecic alopecic aloptia.
4-Niba 4- (3- (4-hydroxybutyl) -4,4-dimethyl-2,5-dioxo-1-midazoromethyl) Bengenitrile yumwuka mwiza;Mugihe cyo guhuza uruhu, ukure imyenda yanduye, uruhu rwuzuye hamwe nisabune namazi, kandi ushake ubuvuzi niba bitameze neza;
Ingaruka
Ru58841 ikoreshwa kumutwe, yinjijwe numusatsi wabisebe, kandi mubyukuri, irashobora kwinjiza amaraso kandi ikagira ingaruka kubindi bice byumubiri. Ariko nta ngaruka zifatika zabonetse mubushakashatsi bwibisabwa byibanze mu nguge. Ariko, abantu bamwe bagerageje Ru58841 bavuga ko bahuye ningaruka zimwe na zimwe ziva mu gukoresha Ru, bagabanaga uruhu, bagabanye inyamanswa, isesemu, isesemi, amaso atukura, azunguruka, kandi afite umutwe.