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Tianeptine Sodium yo kunyura

Ibisobanuro bigufi:

Isura n'imiterere: ikomeye

Ubucucike: 1.38 G / CM3

Gushonga Ingingo: 129-131 ° C.

Ingingo itetse: 609.2ºC kuri 760 MMHG

Flash Ingingo: 322.2ºc

Indangagaciro iroba: 1.639

Kamero: 66981-73-5

MoleCur Fortula: C21H25CLN2O4S

Uburemere bwa molekile: 436.95200


Ibisobanuro birambuye

Ibicuruzwa

Ibisobanuro birambuye

Izina Tianeptine Sodium
Umubare wa Cas 66981-73-5
Formulala C21h25cln2o4s
Uburemere bwa molekile 436.95200
Gushonga 129-131 ° C.
Ingingo itetse 609.2ºC kuri 760 MMHG
Ubuziranenge 99%
Ububiko Bifunze mu bushyuhe bwumutse, icyumba ubushyuhe
Ifishi Ifu
Ibara Cyera
Gupakira Pe Umufuka + Umufuka wa Aluminium

Synonyme

Tianeptina; Tianeptina [Inn-Icyesipanyoli]; Coaxil; Tianootine; Tianeptum;

Ingaruka ya farumasi

Imikoreshereze

Ahanini ikora kuri sisitemu ya 5-ht, nta byishimo, kwishima, kurwanya acetylcholine na cardiotoxigine. Yo kwiheba.

 

Ingaruka ya farumasi

1. Uburyo bwo kudakunda iki gicuruzwa buratandukanye n'icya TCA gakondo TCA. Irashobora kongera uptake ya 5-ht muri cleft ya synaptic, ariko ifite ingaruka zidakomeye kuri couptake ya 5-ht na na. Birashobora kugira ingaruka zo kuzamura 5-HT Neuronal. Ntabwo ifite isano kubakira m, H1, α1 na α2-na resitora.
2. Ibyifuzo bya antidepression byiki gicuruzwa bisa nibya TCA, numutekano wacyo no kwihanganira biruta TCA (antideprepressique ya Tricyclic). Imikorere yiki gicuruzwa isa niya SSri Fluoxetine.
3. Ubushakashatsi bwibiyobyabwenge bwibiyobyabwenge bwerekanye ko bushobora: Ongera ibikorwa byigihe gito byingirabuzimafatizo za pippocampus hanyuma wihutisha gukira mubikorwa byayo nyuma yo kubuza; Ongera reabsorpription ya 5-hydroxytryptamine na neurons muri contex na hippocampus.

 

Ubushakashatsi Uburozi

- Ibizamini byuburozi, subacute nibizamini byigihe kirekire: Nta mpinduka muri biologiya, imikorere yumwijima, anatory pathologiya.
- Uburozi bwimyororokere nikizamini cya Teratongano: Tianeptine nta ngaruka igira ku bushobozi bw'imyororokere y'ababyeyi bavuwe no ku rubavu n'urubyaro.
- Ikizamini cya mugwage: Tianeptine ntabwo ifite mutasige.


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