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Triamtere cyane cyane uwebwe mugucuruza indwara zidasanzwe

Ibisobanuro bigufi:

Gushonga Ingingo: 316 ° C.

Ingingo itetse: 386.46 ° C (igereranya ribi)

Ubucucike: 1.3215 (rougsesiaiaites)

Indangagaciro irohama: 1.8260 (gendayiza)

Flash Ingingo: 11 ° C.

Imiterere yo kubika: 2-8 ° C.

Gukemurwa: Forticacid: Soluble200mg + 4mlwarmforlicacid, isobanutse, umuhondo-icyatsi

Coeeffity Coeefficient: (PKA) 6.2 (AT25 ℃)

Ibara: ibara ryijimye kumuhondo

Amazi yonyine: <0.1G / 100MLT20000ºC


Ibisobanuro birambuye

Ibicuruzwa

Ibisobanuro birambuye

Izina Triamterene
Umubare wa Cas 396-01-0
Formulala C12H11N7
Uburemere bwa molekile 253.26
Umubare wa EINECS 206-904-3
Ingingo itetse 386.46 ° C.
Ubuziranenge 98%
Ububiko Bifunze mu bushyuhe bwumutse, icyumba ubushyuhe
Ifishi Ifu
Ibara Ibara ry'umuhondo
Gupakira Pe Umufuka + Umufuka wa Aluminium

Synonyme

6-Phenyl-; 7-pteridinetrine, 6-phenyl-4; ditak; ditak; diurene; dyrenium; dytac

Ingaruka ya farumasi

Incamake

Triamterene ni poikesic-paurict, ifite ingaruka za diuretike yo kugumana potasiyumu na sodium isa na spirorolactone, ariko uburyo bwo gukora buratandukanye. Biracyafite ingaruka za diuretic nyuma yo kubuza ibanga rya Aldosterone na sodium chloride cyangwa gukuraho glande ya adrenal. Ahantu hayo hako kuri tubule idahwitse, kubuza kungurana ibitekerezo na podium, potasiyumu, yongera exreque ya Na + no mu nkari, no kugabanya amagambo ya K +. Irashobora kandi kubuza reabsorpription ya NA + no gusohora k + nukusanya duction. Ingaruka ya diuretititic yiki gicuruzwa ni intege nke. Iyo bikoreshejwe hamwe na baluretics nka Thiezide, ntishobora gushimangira ingaruka za kadamu Mubyongeyeho, hariho n'ingaruka zo gusohora aside irike. Gukoresha igihe kirekire birashobora kongera urwego rwa area. Irakoreshwa cyane kuri edema idashidikanywaho cyangwa ascite iterwa no gutsindwa kwumutima, umwijima cirrhose hamwe na nephritis idakira. Irashobora kandi gukoreshwa kubarwayi badakora hamwe na hydrochlorothiazide cyangwa spirorolactone.

 

Ingaruka ya farumasi
Iki gicuruzwa ni poikesic-paurics, kibuza mu buryo butaziguye na + -k + kunguranagura ibituba bya kure no gukusanya imiyoboro ya Na +, Cli-, n'amazi, mu gihe bigabanya expreting ya K +.

 

Ibimenyetso

Irakoreshwa cyane cyane kuvura indwara za edema; Harimo kunanirwa k'umutima, umwijima cirrhosis, syndrome ya nephrotic n'amazi na sodium mugihe cyo kuvura adrenal glucocorticoid ya adrenal glucocorticoid; Irashobora kandi gukoreshwa mugufata Edema ya Idiopathic.

 

Imikoreshereze

Abanyantege nke. Ingaruka zirihuta kandi igihe gito, Diresis itangira amasaha 2 yubuyobozi, igera ku mpinga amasaha 6, kandi ingaruka zimara amasaha 8-12. Ikoreshwa mu buryo bwa edema cyangwa ascite iterwa no kunanirwa k'umutima, umwijima wa cirrhosis hamwe na nephritis idakira, kandi ikoreshwa kuri hydrochlorothiazide cyangwa spirorolacto. imanza. Iki gicuruzwa gifite imikorere yo gukuraho aside irike kandi ibereye kuvura ubwato.

 


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