Izina | Triamterene |
Umubare wa Cas | 396-01-0 |
Formulala | C12H11N7 |
Uburemere bwa molekile | 253.26 |
Umubare wa EINECS | 206-904-3 |
Ingingo itetse | 386.46 ° C. |
Ubuziranenge | 98% |
Ububiko | Bifunze mu bushyuhe bwumutse, icyumba ubushyuhe |
Ifishi | Ifu |
Ibara | Ibara ry'umuhondo |
Gupakira | Pe Umufuka + Umufuka wa Aluminium |
6-Phenyl-; 7-pteridinetrine, 6-phenyl-4; ditak; ditak; diurene; dyrenium; dytac
Incamake
Triamterene ni poikesic-paurict, ifite ingaruka za diuretike yo kugumana potasiyumu na sodium isa na spirorolactone, ariko uburyo bwo gukora buratandukanye. Biracyafite ingaruka za diuretic nyuma yo kubuza ibanga rya Aldosterone na sodium chloride cyangwa gukuraho glande ya adrenal. Ahantu hayo hako kuri tubule idahwitse, kubuza kungurana ibitekerezo na podium, potasiyumu, yongera exreque ya Na + no mu nkari, no kugabanya amagambo ya K +. Irashobora kandi kubuza reabsorpription ya NA + no gusohora k + nukusanya duction. Ingaruka ya diuretititic yiki gicuruzwa ni intege nke. Iyo bikoreshejwe hamwe na baluretics nka Thiezide, ntishobora gushimangira ingaruka za kadamu Mubyongeyeho, hariho n'ingaruka zo gusohora aside irike. Gukoresha igihe kirekire birashobora kongera urwego rwa area. Irakoreshwa cyane kuri edema idashidikanywaho cyangwa ascite iterwa no gutsindwa kwumutima, umwijima cirrhose hamwe na nephritis idakira. Irashobora kandi gukoreshwa kubarwayi badakora hamwe na hydrochlorothiazide cyangwa spirorolactone.
Ingaruka ya farumasi
Iki gicuruzwa ni poikesic-paurics, kibuza mu buryo butaziguye na + -k + kunguranagura ibituba bya kure no gukusanya imiyoboro ya Na +, Cli-, n'amazi, mu gihe bigabanya expreting ya K +.
Ibimenyetso
Irakoreshwa cyane cyane kuvura indwara za edema; Harimo kunanirwa k'umutima, umwijima cirrhosis, syndrome ya nephrotic n'amazi na sodium mugihe cyo kuvura adrenal glucocorticoid ya adrenal glucocorticoid; Irashobora kandi gukoreshwa mugufata Edema ya Idiopathic.
Imikoreshereze
Abanyantege nke. Ingaruka zirihuta kandi igihe gito, Diresis itangira amasaha 2 yubuyobozi, igera ku mpinga amasaha 6, kandi ingaruka zimara amasaha 8-12. Ikoreshwa mu buryo bwa edema cyangwa ascite iterwa no kunanirwa k'umutima, umwijima wa cirrhosis hamwe na nephritis idakira, kandi ikoreshwa kuri hydrochlorothiazide cyangwa spirorolacto. imanza. Iki gicuruzwa gifite imikorere yo gukuraho aside irike kandi ibereye kuvura ubwato.