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Cetrorelix Acetate kugirango irinde intanga ngore 120287-85-6

Ibisobanuro bigufi:

Izina: Cetrorelix acetate

Numero ya CAS: 120287-85-6

Inzira ya molekulari: C70H92ClN17O14

Uburemere bwa molekuline: 1431.04

EINECS Numero: 686-384-6


Ibicuruzwa birambuye

Ibicuruzwa

Ibicuruzwa birambuye

Izina Cetrorelix acetate
Numero ya CAS 120287-85-6
Inzira ya molekulari C70H92ClN17O14
Uburemere bwa molekile 1431.04
Umubare wa EINECS 686-384-6

Synonyme

AC- (D-ALA [3- (2-NAPHTHYL)]) - [D-PHE (4-CL)] - (D-ALA [3- RG-PRO-D-ALA-OH; Cetrorelixacetate; CETRORELIX; CETRORELIXACID; CETRIZINEDIHYDROCHLORIDE; C; hemicalbookN-Acetyl-3- (2-naphthalenyl) -D-Ala-4-chloro-D-Phe-3- (3-pyridyl) -D-Ala-L-Ser-L-Tyr-N5- (aminocarbonyl) -D-Orn-L-Leu-L-Arro-L-Pro-D-Ala;

Ibisobanuro

Cetrorelix acetate ni decapeptide ya syntetique, ikoreshwa cyane cyane mu buhanga bw’imyororokere ifasha mu gukumira intanga ngore ku barwayi bafite intanga ngore. Ni antagonist ya gonadotropine irekura (GnRH) ishobora guhangana na endogenous LHRH kugirango ihuze reseptors kuri membrane ya pitoito, bityo bikabuza gusohora imisemburo ya luteinizing (LH) hamwe na misemburo itera imisemburo (FSH) na pitoito muburyo butandukanye.

Cetrorelix acetate ni imisemburo ya gonadotropine irekura (GnRH) antagonist. Iki gicuruzwa kirushanwa na endogenous GnRH kubakira ku ngirabuzimafatizo ya pitoito, bityo bikabuza gusohora imisemburo ya endogenous luteinizing (LH) hamwe na hormone itera imisemburo (FSH), bigatinda kugaragara kw'impinga ya LH, bityo bikagenzura intanga ngabo. Ingaruka yiki gicuruzwa ni dose-biterwa, ingaruka zo kubuza ziraziguye, kandi zikomezwa no kuvurwa ubudahwema, nta gutera kwiyongera kwambere mubikorwa bya reseptor ya progesterone bikurikirwa no kugabanuka.

Ibikoresho biva mu ishami rishinzwe ubuziranenge

Amashanyarazi yubushyuhe bwamazi yamashanyarazi

Agasanduku k'ubwoko bw'isanduku

Gushyushya amashanyarazi guhora ubushyuhe bwumye

Ubushyuhe

Isesengura ry'utugingo ngengabuzima

Amazi ya chromatografiya

Polarimeteri yikora

Imirasire

UV / Ifoto igaragara

Agasanduku ko kumisha amashanyarazi

Umuvuduko ukabije wa parike sterilizer

Metero ya PH

Ikizamini gisobanutse

Ikizamini cya Osmolality

Isesengura rya Cassette

Isesengura ryinshi

Agasanduku ko kumashanyarazi

Biochemical incubator

Inkubator

Aseptic izigunga

Ikoreshwa rya karubone yose

Ibiro byumye

Icyumba cyo gupima ibiyobyabwenge byuzuye

Ubushyuhe burigihe hamwe no kwiyuhagira amazi

Agasanduku ko kubika firigo

Gas Chromatograf

Inama y’umutekano y’ibinyabuzima

Intebe isukuye

TOC hamwe nuyobora

TOC hamwe nuburyo bwiza bwo gutanga no kugaruka bikurikiranwa buri gihe. TOC ikurikiranwa na QC buri cyumweru. Imikorere ikurikiranwa kumurongo kandi ikandikwa nuwashinzwe amazi meza asukuye rimwe mumasaha ane. Imikorere ikurikiranwa kuri RO ibanza, RO yisumbuye, EDI hamwe nibisubizo byose byo kugabura sisitemu. Ibisobanuro by'amazi meza birahari kandi bihuye nibisobanuro byateganijwe mbere bitarenze 1.3 µs / cm kuri 25 ° C (USP). Kubintu nyamukuru byo gutanga no kugaruka, ikizamini cyuzuye. ikorwa buri cyumweru, kubindi ukoresheje ingingo mukuzenguruka, ikizamini cyuzuye gikorwa rimwe mukwezi. Ikizamini cyuzuye kirimo inyuguti, pH, nitrate, nitrite, ammonia, imiyoboro, TOC, ibintu bidahindagurika, ibyuma biremereye, imipaka ya mikorobe na endotoxine ya bagiteri.


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